This paper proposes an efficient envelope delta-sigma based transmitter architecture with gate bias modulation for modern wireless communication systems. Using this architecture, envelope varying signals are converted to constant envelope signals. The constant envelope phase signal is up-converted and amplified utilizing high efficiency power amplifier, while the two level delta-sigma modulated envelope signal is used to switch the gate of the power amplifier. To validate the proposed technique, a prototype transmitter is implemented and evaluated. A Long-Term Evolution (LTE) uplink signal with the bandwidth of 3.84 MHz and the peak-to average power ratio (PAPR) of 7 dB is used to validate the linearity and efficiency performance of the transmitter setup. Using the LTE uplink signal, the polar architecture with modulated gate bias is able to achieve the average drain efficiency of 48% and PAE of 42% at the output power of 25.5dBm. The adjacent channel leakage ratio (ACLR) measured for this signal is less than −31dBc at 10 MHz offset from the center frequency of 2.35GHz. The measurement results are able to meet the spectrum mask without linearization techniques.